CAS NO: | 362665-57-4 |
包装 | 价格(元) |
10mg | 电议 |
50mg | 电议 |
产品名称: | 替洛利生草酸盐 |
CAS: | 362665-57-4 |
分子式: | C19H28ClNO5 |
分子量: | 385.88 |
纯度: | >98% |
溶解性: | DMSO |
存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months; -20℃ 1 month |
研究领域: | Neurological Disease |
Target: | Ki: 0.16 nM (H3 receptor)[1];EC50: 1.5 nM (H3 receptor)[1] |
描述: | Pitolisant oxalate is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). |