CAS NO: | 1802175-07-0 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
CAS: | 1802175-07-0 |
分子式: | C27H36N4O5S |
分子量: | 528.66 |
纯度: | ≥98% |
溶解性: | DMSO |
存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
研究领域: | Cancer |
Target: | IC50: 0.24 nM (EZH2 WT), 0.51 nM (EZH2 Y641N), 6.1 nM (EZH1) |
描述: | CPI-169 is a novel and potent EZH2 inhibitor, with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively. |