CAS NO: | 1015787-98-0 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
CAS: | 1015787-98-0 |
分子式: | C14H19N5O4S |
分子量: | 353.40 |
纯度: | >98% |
溶解性: | DMSO : 5 mg/mL (14.15 mM; ultrasonic and adjust pH to 5-6 with HCl) |
存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
研究领域: | Inflammation/Immunology |
Target: | IC50: ~30 nM (recombinant hP2X3 homotrimers), 100-250 nM (hP2X2/3 heterotrimeric receptors) |
描述: | Gefapixant is an orally active P2X3 receptor (P2X3R) antagonist with IC 50s of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. |