Methyl-6-alpha-Naltrexol 是甲基纳曲酮 (MNTX) 的代谢物 (metabolite)。Methyl-6-alpha-Naltrexol 是一种选择性的 mu-阿片受体 (mu-opioid receptor) 拮抗剂，在胃肠道组织中起外周作用的受体拮抗剂作用。
货号:ajcx34964
CAS:116388-85-3
分子式:C21H27NO4
分子量：357.44
溶解度:N/A
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Methyl-6-alpha-Naltrexol is a metabolite of Methylnaltrexone (MNTX). Methylnaltrexone is a selective mu-opioid receptor antagonist and functions as a peripherally acting receptor antagonist in tissues of the gastrointestinal tract[1].

[1]. Appavu Chandrasekaran,et al. Metabolism of intravenous methylnaltrexone in mice, rats, dogs, and humans. Drug Metab Dispos. 2010 Apr;38(4):606-16.