8-Cyclopentyl-1,3-dimethylxanthine (Compound 2a) 是一种选择性腺苷 A1 受体拮抗剂，对 A1 受体和 A2 受体的 Kis 分别为 10.9 nM 和 1440 nM。
货号:ajcx27402
CAS:35873-49-5
分子式:C12H16N4O2
分子量：248.28
溶解度:DMF: 1 mg/ml,DMSO:PBS (pH 7.2) (1:20): 0.04 mg/ml
纯度：98%
存储：Store at -20°C
库存：现货

Background:

High affinity adenosine A1 receptor antagonist (pKi = 7.5-8).

Dalpiaz et al (1998) Thermodynamics of full agonist, partial agonist, and antagonist binding to wild-type and mutant adenosine A1 receptors. Biochem.Pharmacol. 56 1437 PMID:9827575