CAS NO: | 1245907-03-2 |
规格: | 98% |
分子量: | 392.93 |
包装 | 价格(元) |
10mg | 电议 |
50mg | 电议 |
Background:
Potent Aurora kinase A inhibitor (Ki = 1.2 nM compared to 101 nM for inhibition of Aurora kinase B). Selective over 60 other kinases (IC50 values >1000 nM). Exhibits good cell permeability and antitumor activity.