RSK2-IN-2 (Compound 25) 是 RPS6KA3 (RSK2) 激酶的可逆共价抑制剂。 RSK2-IN-2 也抑制MSK1、MSK2和RSK3。

RSK2-IN-2 (Compound 25) is a reversible covalent inhibitor of the RPS6KA3 ( RSK2 ) kinase. RSK2-IN-2 is also described to inhibit MSK1, MSK2 and RSK3 [1].

RSK2-IN-2 (Compound 25) shows strong activity with ERK2-MSK1 cascade pIC 50 of 9.6 [1].

1637749-78-0

C16H11N5O

289.29

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years